Tracleer
Generic Name:
Bosentan
Brand Names:
Tracleer
Tracleer Description:
Tracleer is an endothelin receptor antagonist prescribed to treat pulmonary arterial hypertension (PAH), a condition involving high blood pressure in the blood vessels of the lungs. Tracleer helps to relax the blood vessels in the lungs by blocking a particular hormone, which allows blood to flow more easily and improves a patient's ability to exercise.
Tracleer Side Effects:
Tracleer has been linked to the following serious side effects:
- Birth defects
- Liver damage
- Low red blood cell count (anemia)
- Reduced sperm count
For more information, see Tracleer side effects page.
Tracleer Uses:
Tracleer is prescribed to treat pulmonary arterial hypertension (PAH), a condition which can cause the following symptoms:
- Shortness of breath
- Dizziness
- Tiredness
Tracleer may help improve the ability to exercise in patients with PAH, as well as slow down the worsening of a patient's physical condition.
Tracleer Interactions:
Tell your doctor about all prescription and non-prescription medications you may be taking along with Tracleer, including vitamins, nutritional supplements, and herbal products. The following drugs may interact with this medication:
- Blood thinners such as warfarin (Coumadin)
- Cyclosporine A
- Glyburide
- Hormone-based forms of birth control, such as oral contraceptives, birth control patches, shots, or implants (they may be ineffective)
- Ketoconazole, fluconazole, itraconazole, and voriconazole
- Lopinavir, ritonavir, atazanavir, darunavir, fosamprenavir, saquinavir, tipranavir, or other HIV medications
- Rifampin
- Sildenafil
- Simvastatin, lovastatin, atorvastatin, and other "-statin" medications for high cholesterol
- Tacrolimus
Tracleer Dosage Information:
Typical Dosage Recommendations
Tracleer dosages may vary among patients. Your doctor will establish the size and frequency of your dosage according to your individual needs. It is important to follow the guidelines established by your doctor.
Tracleer is generally prescribed to be taken as 62.5 mg twice daily for 4 weeks. Dosage may be gradually increased, if needed, to 125 mg twice daily. Tracleer should be given in the morning and evening, with or without food.
Missing a Dose of Tracleer
If you miss a dose of Tracleer, take the missed dose as soon as you remember. If it is almost time for your next scheduled dose, skip the missed dose and wait to return to your regular dosing schedule.
Tracleer Overdose
Seek emergency medical attention if you think you have used too much of this medication. Signs of overdose include headache, upset stomach, vomiting, fast heartbeat, fainting, dizziness, and blurred vision.
Tracleer FDA Approval:
November 20, 2001
Tracleer Recall/Black Box Warning Information:
There is a Black Box warning on Tracleer concerning the serious risks of liver problems and birth defects associated with the medication. Patients are required to schedule monthly liver function tests and pregnancy tests during treatment with Tracleer.
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September 7, 2010, 9:59 am
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September 2, 2010, 12:51 pm
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September 1, 2010, 3:16 pm
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August 31, 2010, 2:01 pm
